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Publication
PropertyValue
Working Groups RG Griesinger, RG de Groot
SubprojectNone
Open AccessOpen Access Yes
Publication TypePreprint
Peer ReviewedNo
DOIDOI 10.1101/2025.05.30.655790
Publication Year2025
TitleThe clinical drug candidate anle138b binds predominantly to the central cavity in lipidic Aβ₄₀ fibrils and modulates fibril formation
JournalbioRxiv
ISSNno ISSN (NLM ID:101680187)
URL https://doi.org/10.1101/2025.05.30.655790
Journal AbbreviationbioRxiv
AuthorsHan M, Frieg B, Matthes D, Leonov A, Ryazanov S, Giller K, Nimerovsky E, Stampolaki M, Xue K, Overkamp K, Dienemann C, Riedel D, Giese A, Becker S, de Groot BL, Schröder GF, Andreas LB, Griesinger C
First AuthorHan M
Last AuthorGriesinger C

 External Resources

 biorxiv....ll.pdf  Article fulltext

 53129  BMRB identifier (53129)

 NCT04685265  ClinicalTrials ID (NCT04685265, reused)

 NCT06568237  ClinicalTrials ID (NCT06568237, reused)

 10.17617/3.NRYUVQ  DOI (10.17617/3.NRYUVQ, Edmond, does not yet resolve)

 EMD-53880  EMBL-EBI EMDB identifier (EMD-53880)

 EMD-53882  EMBL-EBI EMDB identifier (EMD-53882)

 44608289  NCBI PubChem (44608289, Emrusolmin)

 0009-0004-8007-5711  ORCID identifier (Mookyoung Han)

 0000-0002-7877-0262  ORCID identifier (Benedikt Frieg)

 0000-0003-3969-6335  ORCID identifier (Dirk Matthes)

 0000-0002-5586-9382  ORCID identifier (Andrei Leonov)

 0000-0002-4149-7899  ORCID identifier (Karin Giller)

 0000-0003-3002-0718  ORCID identifier (Evgeny Nimerovsky)

 0000-0002-0144-4792  ORCID identifier (Marianna Stampolaki)

 0000-0002-2172-5110  ORCID identifier (Christian Dienemann)

 0000-0003-2970-6894  ORCID identifier (Dietmar Riedel)

 0000-0002-8238-4102  ORCID identifier (Armin Giese)

 0000-0003-2041-5740  ORCID identifier (Stefan Becker)

 0000-0003-3570-3534  ORCID identifier (Bert L. de Groot)

 0000-0003-1803-5431  ORCID identifier (Gunnar F. Schröder)

 0000-0003-3216-9065  ORCID identifier (Loren B. Andreas)

 0000-0002-1266-4344  ORCID identifier (Christian Griesinger)

 9RAW  RCSB PDB Identifier (DOI:10.2210/pdb9RAW/pdb)

 9RAX  RCSB PDB Identifier (DOI:10.2210/pdb9RAX/pdb)

 8ovk  RCSB PDB Identifier (DOI:10.2210/pdb8ovk/pdb, reused)

 02nv7yv05  ROR identifier (02nv7yv05, Forschungszentrum Jülich)

 024z2rq82  ROR identifier (024z2rq82, Heinrich Heine University Düsseldorf)

 03av75f26  ROR identifier (03av75f26, Max Planck Institute for Multidisciplinary Sciences)

 05xy1nn52  ROR identifier (05xy1nn52, Multiscale Bioimaging)

 SCR_014222  SciCrunch identifier (RRID:SCR_014222, Coot)

 SCR_018392  SciCrunch identifier (RRID:SCR_018392, crYOLO)

 SCR_016732  SciCrunch identifier (RRID:SCR_016732, CTFFIND)

 SCR_008619  SciCrunch identifier (RRID:SCR_008619, Gnuplot)

 SCR_014565  SciCrunch identifier (RRID:SCR_014565, GROMACS)

 SCR_014479  SciCrunch identifier (RRID:SCR_014479, Inkscape)

 SCR_016137  SciCrunch identifier (RRID:SCR_016137, Microsoft Excel)

 SCR_014226  SciCrunch identifier (RRID:SCR_014226, MolProbity)

 SCR_014224  SciCrunch identifier (RRID:SCR_014224, Phenix)

 SCR_000305  SciCrunch identifier (RRID:SCR_000305, PyMOL)

 SCR_008394  SciCrunch identifier (RRID:SCR_008394, Python)

 SCR_016274  SciCrunch identifier (RRID:SCR_016274, RELION)

 SCR_015872  SciCrunch identifier (RRID:SCR_015872, UCSF ChimeraX)

 mbexc.de...ation/  Website entry (mbexc.de)